许庆龙,男,中国药科大学新药研究中心特聘研究员,博士生导师。2007年毕业于安徽师范大学化学系获学士学位(应用化学);2012年获中国科学院上海有机化学研究所博士学位(有机化学);2012-2014年在美国西南医学研究中心从事博士后研究。主要从事有机合成化学和新药导向的方法学研究,在SCI核心期刊JACSAngewScience等发表论文10余篇。

主持课题

1)高级人才引进项目1项;

2)国家自然科学基金青年项目1项;

3)江苏省自然科学基金青年项目1项。

近期发表论文:

1. Peng-Fei Wang, Chun-Huan Jiang, Xiaoan Wen, Qing-Long Xu* and Hongbin Sun*; C–H Bond Functionalization via [1,5]-Hydride Shift/Cyclization Sequence: Approach to Spiroindolenines. J. Org. Chem. 2015, 80, 1155-1162. (IF 4.721)

2. Xiantao Lei, Chun-Huan Jiang, Xiaoan Wen, Qing-Long Xu* and Hongbin Sun*; Formal [4+1] cycloaddition of o-quinone methides: facile synthesis of dihydrobenzofurans. RSC Adv. 2015, 5, 14953-14957. (IF 3.840)

3. Le Zhen, Chao Lin, Hong-Jin Du, Liang Dai, Xiaoan Wen, Qing-Long Xu* and Hongbin Sun*; Quinone Methides as [1, 5]-Hydride Acceptors: Approach to N-Aryl Pyrroles. Tetrahedron 2015, 71, 2839-2843. (IF 2.641)

4. Fan Zhang, Hengzhi Sun, Zhuang Song, Shuxi Zhou, Xiaoan Wen, Qing-Long Xu* and Hongbin Sun*; Stereoselective Synthesis of Arylglycine Derivatives via Palladium-Catalyzed α-Arylation of a Chiral Nickel(II) Glycinate. J. Org. Chem. 2015, 80, 4459–4464. (IF 4.721)

5. Xiantao Lei, Hong-Yan Xie, Si-Yuan Chen, Kai-Shun Teng, Xiaoan Wen, Qing-Long Xu* and Hongbin Sun*; Approach to N-aryl pyrroles via diphenyl phosphate-catalyzed [1,5]-Hydride shift/isomerization reaction with indoles. Tetrahedron 2015, 71, 4098-4101. (IF 2.641)

6. Chao Lin, Le Zhen, Yong Cheng, Hong-Jin Du, Hui Zhao, Xiaoan Wen, Ling-Yi Kong, Qing-Long Xu* and Hongbin Sun*; Visible-Light Induced Isoindoles Formation To Trigger Intermolecular Diels–Alder Reactions in the Presence of Air. Org. Lett. 2015, 17, 2684-2687. (IF 6.364)

7. Yong-Zhi Chang, Ming-Lei Li, Wen-Feng Zhao, Xiaoan Wen, Hongbin Sun,*and Qing-Long Xu*; Construction of Oxadiazepines via Lewis Acid-Catalyzed Tandem 1,5-Hydride Shift/Cyclization. J. Org. Chem. 2015, 80, 9620–9627. (IF 4.721)

8. Peng-Fei Wang, Ya-Ping Huang, Xiaoan Wen, Hongbin Sun,* and Qing-Long Xu*; Concise Access to 1,2-Pyrrole-Annulated Benzazepines through a Brønsted Acid Catalyzed Redox-Neutral Domino Reaction. Eur. J. Org. Chem. 2015, 6727–6733. (IF 3.065)

9. Hongyin Gao, Qing-Long Xu, (共同一作) Craig Keene, Muhammed Yousufuddin, Daniel H. Ess, László Kürti*; Practical Organocatalytic Synthesis of Non-C2-Symmetrical Atropoisomeric BINOL/NOBIN-Type Functionalized Biaryls. Angew. Chem. Int. Ed. 2015, 54, DOI: 10.1002/anie.201508419. (IF 11.261)

10. Zheng-Le Zhao, Qing-Long Xu, Qing Gu, Xin-Yan Wu* and Shu-Li You*; Enantioselective synthesis of 4-substituted tetrahydroisoquinolines via palladium-catalyzed intramolecular Friedel–Crafts type allylic alkylation of phenols. Org. Biomol. Chem. 2015, 13, 3086-3092. (IF 3.562)

11. Asymmetric Functionalization of C-H Bonds, 8,9章, 2015.10RSC Publishing

12. Fan Zhang, Xiaoan Wen, Qing-Long Xu* and Hongbin Sun*; Asymmetric Synthesis of 3,4-Disubstituted Proline Derivatives: Application in Synthesis of Hepatitis C Virus Protease Inhibitor Telaprevir. Eur. J. Org. Chem. 2014, 8101–8109. (IF 3.154)

13. Hong-Jin Du, Le Zhen, Xiaoan Wen, Qing-Long Xu* and Hongbin Sun*; Intramolecular redox reaction for the synthesis of N-aryl pyrroles catalyzed by Lewis acids. Org. Biomol. Chem. 2014, 12, 9716-9719. (IF 3.487)

14. Chun-Huan Jiang, Xiantao Lei, Le Zhen, Hong-Jin Du, Xiaoan Wen, Qing-Long Xu* and Hongbin Sun*; Lewis acid-catalyzed redox-neutral amination of 2-(3-pyrroline-1-yl)benzaldehydes via intramolecular [1,5]-hydride shift/isomerization reaction. Beilstein J. Org. Chem. 2014, 10, 2892–2896. (IF 2.803)

15. Hongyin Gao, Qing-Long Xu, Muhammed Yousufuddin, Daniel Halsell Ess, László Kürti*; Low-Temperature, Transition-Metal-Free Intramolecular Amination of Arene C-H Bonds: Rapid Synthesis of Fused N-Heterocycles. Angew. Chem., Int. Ed. 2014, 53, 2701. (IF 11.336)

16. Hongyin Gao, Qing-Long Xu, Craig Keene, László Kürti*; Scalable, Transition-Metal-Free Direct Oxime O-Arylation: Rapid Access to O-Arylhydroxylamines and Substituted Benzo[b]furans. Chem. Eur. J. 2014, 20, 8883. (IF 5.696)

17. Jawahar L. Jat, Mahesh P. Paudyal, Hongyin Gao, Qing-Long Xu, Muhammed Yousufuddin, Deepa Devarajan, Daniel H. Ess*, László Kürti*, John R. Falck*; Direct Aziridination of Olefins: Stereospecific Synthesis of N-H/N-Me Aziridines. Science, 2014, 343, 61. (IF 31.477)

18. 赖增伟,徐黎,宋壮,雷显涛,许庆龙*,孙宏斌*。西他沙星关键中间体胺基氮杂螺环的不对称合成研究。中国药科大学学报201445400-404

19. Qing-Long Xu, Wen-Bo Liu, Li-Xin Dai, Shu-Li You*; Ir-Catalyzed Enantioselective Allylic Substitution of O-Allyl Carbamothioates. J. Org. Chem. 2010, 75, 4615. (IF 4.721)

20. Qing-Long Xu, Li-Xin Dai, Shu-Li You*; Tandem Ir-Catalyzed Allylic Substitution Reaction of Allyl Sulfinates and Isomerization. Org. Lett. 2010, 12, 800. (IF 6.364)

21. Qing-Long Xu, Li-Xin Dai, Shu-Li You*; Enantioselective Synthesis of Tetrahydroisoquinolines via Iridium-Catalyzed Intramolecular Friedel-Crafts- Type Allylic Alkylation of Phenols. Org. Lett. 2012, 14, 2579. (IF 6.364)

22. Qing-Long Xu, Li-Xin Dai, Shu-Li You*; Iridium-Catalyzed Enantioselective Allylic Alkylation of Methyl 2-(4-nitrophenylsulfonyl)acetate and Subsequent Transformations. Adv. Synth. Catal. 2012, 354, 2275. (IF 5.663)

23. Qing-Long Xu, Li-Xin Dai, Shu-Li You*; Diversity Oriented Synthesis of Indole-based Peri-annulated Compounds via Allylic Alkylation Reactions. Chem. Sci. 2013, 4, 97. (IF 9.221)

24. Qing-Long Xu, Hongyin Gao, Muhammed Yousufuddin, Daniel Halsell Ess, László Kürti*; Aerobic, Transition-Metal-Free, Direct and Regiospecific Mono-α-Arylation of Ketones: Synthesis and Mechanism by DFT Calculations. J. Am. Soc. Chem. 2013, 135, 14048. (IF 12.113)

25. Qing-Long Xu, Chun-Xiang Zhuo, Li-Xin Dai, Shu-Li You*; Highly Enantioselective Synthesis of Tetrahydrocarbolines via Iridium-Catalyzed Intramolecular Friedel–Crafts Type Allylic Alkylation Reactions. Org. Lett. 2013, 15, 5909. (IF 6.364)

26. Zhen Feng, Qing-Long Xu, Li-Xin Dai, Shu-Li You*; Enantioselective Synthesis of 2-Aryl-2,3-dihydro-4-quinolones by Chiral Brønsted Acid Catalyzed Intramolecular Aza-Michael Addition Reaction. Heterocycles 2010, 80, 765. (IF 1.079)

27. Zhen Feng, Mi Zeng, Qing-Long Xu, Shu-Li You*; Asymmetric Intramolecular Oxa-Michael Addition of Activated α,β-Unsaturated Ketones by Chiral N-Triflyl Phosphoramide. Chin. Sci. Bull. 2010, 55, 1723. (IF 1.579)

28. Chun-Xiang Zhuo, Qing-Feng Wu, Qiang Zhao, Qing-Long Xu, Shu-Li You*; Enantioselective Functionalization of Indoles and Pyrroles via an In-situ Formed Spiro Intermediate. J. Am. Soc.Chem. 2013, 135, 8169. (IF 12.113)

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